Clenbuterol and Ketotifen best results!

How to use Ketotifen

No Comments

How to use Ketotifen



Introduction Ketotifen Sopharma


I see a lot of newbies trying to find information on Ketotifen so I thought it would be best to put it all together in one post. I gathered this information from a wide range of trusted sources and added my own experiences too. Ketotifen truly is a wonder drug for bodybuilding.

What Is It Ketotifen Sopharma?

Ketotifen is very safe antihistamine used extensively in Europe to treat bronchial asthma and allergies. It is also being studied as a treatment for colitis. When used for asthma, weight gain and an increase in appetite are among the most frequent side effects. Ketotifen also protects the cells in the stomach, small intestine and perhaps the rest of the gut from a number of toxins. A number of case studies suggest that it may be helpful treating skin problems such as acne. Ketotifen also reduces edema (swelling and puffiness caused by water retention) around sores.

Ketotifen Sopharma Studies

German researchers have published data showing that ketotifen lowers TNF-Alpha in the test tube. One study used ketotifen in combination with Oxymethalone, a steroid which helps people gain weight, so it is hard to gauge what effect ketotifen had (the study notes a 14% reduction in TNF-Alpha levels and weight gains of 11-12 pounds in less than four weeks). A larger placebo controlled study of this combination is underway. The other study used ketotifen by itself in eight patients with elevated TNF-alpha, (but no wasting). Taking ketotifen for 12 weeks, these patients gained an average of six pounds, had increases in their body cell mass and reductions in their TNF-alpha levels.

Side Effects and Toxicity

Ketotifen is virtually non-toxic (although it is not advised for patients with epilepsy). People who took twenty times the recommended dose (in suicide attempts) suffered no serious consequences (other than embarrassment). Its primary side effects seem to be temporary drowsiness, dry mouth,(and other mucous membranes) appetite stimulation and weight gain.

Dosing and Side-Effects

No studies have been completed to find the most effective dose but the German researchers used 4 mg daily. Dan Duchaine (who discovered Ketotifen’s use for bodybuilding) suggested 10mg daily but in my experience this is too much and is not beneficial as it makes you far too sleepy. I find that 3-4mg daily seems ideal. However, much higher doses have been shown to be quite safe with no adverse affects other than increased drowsiness and appetite – it will make you hungry for solid food. You can split the dose throughout the day or take it all at once, it doesn’t really matter.

Ketotifen Sopharma and Clenbuterol Sopharma


Clenbuterol is a beta 2 agonist which has a limited anabolic effect during its first few days of use and afterward is normally used to fight fat. At higher doses, however, it can be catabolic to muscle and it must be cycled on a 2 week on, 2 week of basis or the beta 2 receptors that clenbuterol binds to become saturated and down regulate.
Ketotifen’s magic is that it upregulates the beta-receptors including the beta 2’s that clen uses. As long as you are taking ketotifen, it will continue to clean these receptors, meaning they will not downregulate – even while on a heavy clen cycle. That means you can continue to take clen indefinitely without having to cycle off to regenerate the receptors. 2-3mg daily can upregulate even severely shut down receptors within a week.
It also means that you don’t need as much clenbuterol to get the same benefits. You can take about 30-40% less clenbuterol and it will be equally as effective. It also increases the number of receptor sites on the surface of the cell, allowing more clenbuterol to attach, perhaps this is the reason for the increased efficiency. Ketotifen also seems to lessen the sides of clenbuterol, including the jitters.
For a thorough guide on how to use clenbuterol, make sure to check out:
How to Use Clenbuterol Effectively to Speed up Fat-Loss

Ketotifen Sopharma and ECA

Perhaps an even better use for ketotifen is taking it with the ECA stack. While the thermogenic effect of ephedrine is not as potent as clen because it doesn’t have a high receptor affinity, and it is not limited to beta-2 receptors. In fact it seems to have a good effect on beta 3 receptors as well, which act as a type of thermogenic messenger and over half of ephedrine effect is from beta-3 stimulation. Clen has almost no effect on beta 3 however. So by keeping the beta 2 receptors up, ketotifen can allow the benefits of continuous beta 2 and beta 3 stimulation from ephedrine.

Leave a Reply

Your email address will not be published. Required fields are marked *

Recent Posts

In terms of a dosing schedule for clenbuterol, most users would be well served to split their dosages into two or three evenly spaced doses throughout the day. The first can be taken upon rising and then the one or two others throughout the rest of the morning and/or afternoon.     This is due […]

Where to Look For Clenbuterol

Where to Look For Clenbuterol Online   In this post, we will try to give you some guidance on where to look for clenbuterol deals online. There are several websites that provide information on how to buy clenbuterol, but the tips we’ll offer are very valuable and need to be taken into consideration:   1. […]

Clenbuterol Buy Sale

Clenbuterol Buy Sale with PayPal   There have been many questions on the web on how to buy clenbuterol with PayPal. So far, i have not seen or heard anyone offering PayPal payments for clenbuterol orders. There might be some online shops that offer PayPal payments, but you need to be aware of the following: […]

Clenbuterol Side Effects

Clenbuterol Side Effects You Must Know   People take Clenbuterol for several different reasons however the two primary reasons they drive them aren’t why it had been intended to begin with. This specific drug was produced to be able to help individuals with bronchial asthma also it is a kind of steroid. The unfortunate factor […]

Ideal Dosage for Clenbuterol Cycle

Ideal Dosage for Clenbuterol Cycle   The Clenbuterol cycle assists those body builders who have a two day on as well as a two day off fitness regime. They other cycle used for this performance enhancing drug is that of a three week on three week off body building regime. Supplements such as Taurine and […]

Buying Clenbuterol Shopping Store Guide

Buying Clenbuterol Shopping Store Guide   There have been many websites offering clenbuterol on the internet. People usually wonder around and not sure from which one to buy. We have created the blog “Buying Clenbuterol” in order to digg in and research on the buying process of clenbuterol. Our research and analysis will be shared […]